Biotinylated kinases are now available from Carna Biosciences. These important reagents are best suited for the study of binding affinity and other kinase-molecule interactions on devices measuring Surface Plasmon Resonance (SPR), BioLayer Interferometry (BLI) and other similar values. They can also be utilized in homogenous proximity-based binding assays such as TR-FRET to interrogate inhibitor binding affinity, determine on-off rates, and measure binding kinetics.
The immobilization of target proteins onto sensor surfaces without impairing their structure and activity can be quite a challenging step in small molecule drug discovery.
Carna' s in-house single-site specifically biotinylated kinases can easily facilitate this immobilization and lead to the acquisition of real-time and accurate data for quick evaluation in your programs.
Advantages vs. Chemical Biotinylation
Some Biotinylated Protein products are pre-activated with ATP treatment (indicated with *). For those products, we provide ”non-activated” version without ATP treatment in the production process (some still in production). Those can be useful for binding analysis between your target kinase in an inactive form and your compound.
Product | Cat.No. | Storage | PKG Size | Price(US$) | |
---|---|---|---|---|---|
BTN - ABL(ABL1), Length: Full-length | 08-401-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - ABL(ABL1), Length: Full-length | 08-401-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - ACTR2B(ACVR2B), Length: Cytoplasmic domain | 09-432-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - ACTR2B(ACVR2B), Length: Cytoplasmic domain | 09-432-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - AKT1, Length: Catalytic domain | 01-401-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - AKT1, Length: Catalytic domain | 01-401-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - AKT2, Length: Catalytic domain | 01-402-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - AKT2, Length: Catalytic domain | 01-402-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - ALK, Length: Cytoplasmic domain | 08-405-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - ALK, Length: Cytoplasmic domain | 08-405-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - ALK[L1196M], Length: Cytoplasmic domain | 08-429-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - ALK[L1196M], Length: Cytoplasmic domain | 08-429-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - AurA(AURKA), Length: Full-length | 05-401-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - AurA(AURKA), Length: Full-length | 05-401-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN-AurB(AURKB)/INCENP, Length: Full-length | 05-402-21N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN-AurB(AURKB)/INCENP, Length: Full-length | 05-402-21N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - AXL, Length: Cytoplasmic domain | 08-407-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - AXL, Length: Cytoplasmic domain | 08-407-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - BMX, Length: Full-length | 08-479-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - BMX, Length: Full-length | 08-479-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - BTK, Length: Full-length | 08-480-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - BTK, Length: Full-length | 08-480-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN-BTK[non-activated], Length: Full-length | 08-480-23N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN-BTK[non-activated], Length: Full-length | 08-480-23N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - CHK1(CHEK1), Length: Full-length | 02-417-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - CHK1(CHEK1), Length: Full-length | 02-417-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - DDR2, Length: Cytoplasmic domain | 08-414-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - DDR2, Length: Cytoplasmic domain | 08-414-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - DLK(MAP3K12), Length: Catalytic domain | 09-411-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - DLK(MAP3K12), Length: Catalytic domain | 09-411-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - EGFR, Length: Cytoplasmic domain | 08-415-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - EGFR, Length: Cytoplasmic domain | 08-415-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - EGFR[T790M/L858R], Length: Cytoplasmic domain | 08-410-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - EGFR[T790M/L858R], Length: Cytoplasmic domain | 08-410-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - FAK(PTK2), Length: Truncated protein | 08-437-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - FAK(PTK2), Length: Truncated protein | 08-437-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - FGFR1, Length: Cytoplasmic domain | 08-435-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - FGFR1, Length: Cytoplasmic domain | 08-435-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN-FGFR1 [non-activated], Length: Cytoplasmic domain | 08-435-23N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN-FGFR1 [non-activated], Length: Cytoplasmic domain | 08-435-23N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - FGFR3, Length: Cytoplasmic domain | 08-433-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - FGFR3, Length: Cytoplasmic domain | 08-433-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - FGFR4, Length: Cytoplasmic domain | 08-436-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - FGFR4, Length: Cytoplasmic domain | 08-436-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - FLT3, Length: Cytoplasmic domain | 08-454-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - FLT3, Length: Cytoplasmic domain | 08-454-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - FMS(CSF1R), Length: Cytoplasmic domain | 08-455-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - FMS(CSF1R), Length: Cytoplasmic domain | 08-455-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - FYN[isoform a], Length: Full-length | 08-468-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - FYN[isoform a], Length: Full-length | 08-468-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - IGF1R, Length: Cytoplasmic domain | 08-441-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - IGF1R, Length: Cytoplasmic domain | 08-441-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - IKKb(IKBKB), Length: Truncated protein | 05-484-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - IKKb(IKBKB), Length: Truncated protein | 05-484-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - IKKα(CHUK), Length: Full-length | 05-412-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - IKKα(CHUK), Length: Full-length | 05-412-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - IKKα(CHUK)[inactive mutant], Length: Full-length | 05-412-11-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - IKKα(CHUK)[inactive mutant], Length: Full-length | 05-412-11-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - IRAK4, Length: Full-length | 09-445-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - IRAK4, Length: Full-length | 09-445-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - ITK, Length: Full-length | 08-481-20N-5 | -80°C | 10 µg | 584.00 | Buy |
BTN - ITK, Length: Full-length | 08-481-20N-10 | -80°C | 100 µg | 3,250.00 | Buy |
BTN - JAK1, Length: Catalytic domain | 08-444-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - JAK1, Length: Catalytic domain | 08-444-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - JAK2, Length: Catalytic domain | 08-445-20N-5 | -80°C | 10 µg | 584.00 | Buy |
BTN - JAK2, Length: Catalytic domain | 08-445-20N-10 | -80°C | 100 µg | 3,250.00 | Buy |
BTN - KDR(VEGFR2) , Length: Cytoplasmic domain | 08-491-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - KDR(VEGFR2) , Length: Cytoplasmic domain | 08-491-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - KIT, Length: Cytoplasmic domain | 08-456-21N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - KIT, Length: Cytoplasmic domain | 08-456-21N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - LCK, Length: Full-length | 08-470-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - LCK, Length: Full-length | 08-470-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - LYNa, Length: Full-length | 08-471-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - LYNa, Length: Full-length | 08-471-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - MAP2K1[inactive], Length: Full-length | 07-441-10-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - MAP2K1[inactive], Length: Full-length | 07-441-10-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - MAP3K5, Length: Catalytic domain | 07-407-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - MAP3K5, Length: Catalytic domain | 07-407-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - MET, Length: Cytoplasmic domain | 08-451-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - MET, Length: Cytoplasmic domain | 08-451-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - MNK1(MKNK1), Length: Full-length | 02-445-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - MNK1(MKNK1), Length: Full-length | 02-445-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - NEK9, Length: Truncated protein | 05-433-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - NEK9, Length: Truncated protein | 05-433-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - p38α(MAPK14), Length: Truncated protein | 04-452-20N-5 | -80°C | 10 µg | 584.00 | Buy |
BTN - p38α(MAPK14), Length: Truncated protein | 04-452-20N-10 | -80°C | 100 µg | 3,250.00 | Buy |
BTN - p38α(MAPK14)[inactive], Length: Truncated protein | 04-452-10-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - p38α(MAPK14)[inactive], Length: Truncated protein | 04-452-10-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - PAK4, Length: Full-length | 07-426-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - PAK4, Length: Full-length | 07-426-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - PIK3CA/PIK3R1, Length: Full-length | 11-401-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - PIK3CA/PIK3R1, Length: Full-length | 11-401-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN-PIK3CB/PIK3R1, Length: Full-length | 11-402-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN-PIK3CB/PIK3R1, Length: Full-length | 11-402-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN-PIK3CD/PIK3R1, Length: Full-length | 11-403-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN-PIK3CD/PIK3R1, Length: Full-length | 11-403-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN-PIK3CG, Length: Full-length | 11-404-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN-PIK3CG, Length: Full-length | 11-404-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - PKCη(PRKCH), Length: Full-length | 01-438-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - PKCη(PRKCH), Length: Full-length | 01-438-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - PKN1 , Length: Full-length | 01-444-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - PKN1 , Length: Full-length | 01-444-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - PLK1, Length: Full-length | 05-457-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - PLK1, Length: Full-length | 05-457-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - PYK2(PTK2B), Length: Full-length | 08-438-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - PYK2(PTK2B), Length: Full-length | 08-438-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - RET, Length: Cytoplasmic domain | 08-459-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - RET, Length: Cytoplasmic domain | 08-459-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - ROCK1, Length: Catalytic domain | 01-409-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - ROCK1, Length: Catalytic domain | 01-409-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - SPHK1, Length: Full-length | 11-405-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - SPHK1, Length: Full-length | 11-405-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - SPHK2, Length: Full-length | 11-406-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - SPHK2, Length: Full-length | 11-406-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - SRC, Length: Full-length | 08-473-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - SRC, Length: Full-length | 08-473-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - SRPK1, Length: Full-length | 04-460-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - SRPK1, Length: Full-length | 04-460-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - SYK, Length: Full-length | 08-476-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - SYK, Length: Full-length | 08-476-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN-SYK[non-activated], Length: Full-length | 08-476-23N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN-SYK[non-activated], Length: Full-length | 08-476-23N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN-TAK1-TAB1(MAP3K7), Length: Fused protein | 09-419-21C-5 | -80°C | 10 µg | 449.00 | Buy |
BTN-TAK1-TAB1(MAP3K7), Length: Fused protein | 09-419-21C-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - TGFβR1(TGFBR1), Length: Catalytic domain | 09-441-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - TGFβR1(TGFBR1), Length: Catalytic domain | 09-441-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - TIE2, Length: Cytoplasmic domain | 08-485-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - TIE2, Length: Cytoplasmic domain | 08-485-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - TNIK, Length: Catalytic domain | 07-438-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - TNIK, Length: Catalytic domain | 07-438-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - TRKA(NTRK1), Length: Cytoplasmic domain | 08-486-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - TRKA(NTRK1), Length: Cytoplasmic domain | 08-486-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN-TRKA(NTRK1)[non-activated] , Length: Cytoplasmic domain | 08-486-23N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN-TRKA(NTRK1)[non-activated] , Length: Cytoplasmic domain | 08-486-23N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - TRKB(NTRK2), Length: Cytoplasmic domain | 08-487-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - TRKB(NTRK2), Length: Cytoplasmic domain | 08-487-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN-TRKB(NTRK2)[non-activated], Length: Cytoplasmic domain | 08-487-23N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN-TRKB(NTRK2)[non-activated], Length: Cytoplasmic domain | 08-487-23N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - TRKC(NTRK3), Length: Catalytic domain | 08-497-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - TRKC(NTRK3), Length: Catalytic domain | 08-497-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - TYK2, Length: Catalytic domain | 08-447-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - TYK2, Length: Catalytic domain | 08-447-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |
BTN - WNK1, Length: Catalytic domain | 05-479-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - WNK1, Length: Catalytic domain | 05-479-20N-10 | -80°C | 100 µg | 2,125.00 | Buy |
BTN - WNK4, Length: Catalytic domain | 05-482-20N-5 | -80°C | 10 µg | 449.00 | Buy |
BTN - WNK4, Length: Catalytic domain | 05-482-20N-10 | -80°C | 100 µg | 2,500.00 | Buy |